I-Eprinomectin Injection 1%

Incazelo emfushane:

Ukubukeka: Lo mkhiqizo awunambala ukuya kuketshezi olunamafutha acacile ngokuphuzi, olune-viscous kancane.


Imininingwane Yomkhiqizo

Omaka bomkhiqizo

Incazelo

I-Eprinomectin iyi-abamectin esetshenziswa njenge-endectocide yezilwane. Kuyingxube yezinhlanganisela zamakhemikhali amabili, i-eprinomectin B1a ne-B1b. I-Eprinomectin iwumuthi osebenza kahle kakhulu, obanzi, futhi onensalela ephansi ye-anthelmintic okuwukuphela kwesidakamizwa esine-broad-spectrum anthelmintic esisetshenziswa ezinkomeni zobisi ezincelisayo ngaphandle kwesidingo sokushiywa ubisi futhi ngaphandle kwesidingo sesikhathi sokuphumula.

Eprinomectin

Isimiso Semithi

Imiphumela yocwaningo lwe-kinetic ibonise ukuthi i-acetylaminoavermectin ingamuncwa ngezindlela ezihlukahlukene, njengokujova ngomlomo noma nge-percutaneous, subcutaneous, kanye ne-intramuscular, ngokusebenza kahle kahle nokusabalalisa ngokushesha kuwo wonke umzimba. Kodwa-ke, kuze kube manje, kunamalungiselelo amabili kuphela okuhweba e-acetylaminoavermectin: i-ejenti yokuthulula nomjovo. Phakathi kwabo, ukusetshenziswa kwe-ejenti yokuthulula ezilwaneni ezinonya kulula kakhulu; nakuba i-bioavailability yomjovo iphezulu, ubuhlungu bendawo yomjovo busobala futhi ukuphazamiseka ezilwaneni kukhulu. Kutholwe ukuthi ukumuncwa ngomlomo kungaphezulu kokumuncwa kwe-transdermal ukuze kulawulwe ama-nematode nama-arthropods adla igazi noma uketshezi lomzimba.

Isitoreji

Izakhiwo ze-Physicochemical Umuthi uqinile njengekristale elimhlophe ezingeni lokushisa lasekamelweni, nendawo yokuncibilika engu-173 ° C kanye nokuminyana okungu-1.23 g/cm3. Ngenxa yeqembu layo le-lipophilic esakhiweni salo samangqamuzana, ukuncibilika kwe-lipid kuphezulu, kuncibilika kuzincibilikisi zemvelo ezifana ne-methanol, i-ethanol, i-propylene glycol, i-ethyl acetate, njll., inokuncibilika okukhulu kakhulu ku-propylene glycol (okungaphezu kuka-400 g/ L), futhi cishe ayincibiliki emanzini. I-Eprinomectin kulula ukwenza i-photolyze futhi i-oxidize, futhi into yomuthi kufanele ivikelwe ekukhanyeni futhi igcinwe ngaphansi kwe-vacuum.

Ukusebenzisa

I-Eprinomectin inomphumela omuhle wokulawula ekulawuleni ama-ectoparasites angaphakathi nama-ectoparasites njenge-nematodes, i-hookworms, i-ascaris, i-helminths, izinambuzane nezibungu ezilwaneni ezihlukahlukene ezifana nezinkomo, izimvu, amakamela, nonogwaja. Isetshenziswa kakhulu ekwelapheni i-nematodes yamathumbu, izibungu zokulunywa kanye ne-sarcoptic mange emfuyweni.

Amalungiselelo

Umjovo we-Eprinomectin 1%, i-Eprinomectin Pour-on Solution 0.5%


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